Journal of Natural Sciences Research iiste ISSN 2224-3186 (Paper) ISSN 2225-0921 (Online) Vol.5, No.6, 2015 Design, Synthesis and Acute Anti-Inflammatory Evaluation of New Non-Steroidal Anti-Inflammatory Agents Having 4- Thiazolidinone Pharmacophore Monther F. Mahdi 1 Ayad M. R.Raauf 1 Farah A.H. Kadhim2* 1.Department of Pharmaceutical Chemistry, College of Pharmacy/Al-
Design, Synthesis and in Vivo Anti-inflammatory Activities of 2,4-Diaryl-5-4H-imidazolone Derivatives. Design, synthesis, an d structure-activity relationship for anti-inflammatory drug. Design, Synthesis and In Vitro Evaluation of Novel Anti Title:Design, Synthesis and In Vitro Evaluation of Novel Anti-HIV 3-Pyrazol-3- yl-Pyridin-2-One Analogs VOLUME:15 ISSUE:5 Author(s):Sanjay Kumar, Shiv Gupta, Shraddha Gaikwad, Leila F. Abadi, Late K. K. Bhutani, Smita Kulkarni* and Inder P. Singh* Affiliation:Department of Natural Products, National Institute of Pharmaceutical Education and Research (NIPER), Sector-67, S. A. S. Nagar-160 062
Jan 01, 2020 · Inspired by the promising anti-HBV activity and disclosed structures,, we intend to design, and synthesis new SBAs based on the structure feature of NVR3-778, which were expected to explore structure-activity relationships (SAR) of SBAs, and identify alternative candidate as anti-HBV agents. Download :Download high-res image (132KB) Design, synthesis and biological evaluation of a series of
In search of new and potent anti-ischemic agents, recently we have reported synthesis and biological evaluation of amino-acid based benzodiazepines 8, 9 as new class of anti-ischemic agents (Fig. 1) . However this series of compounds did not exhibit very good potency in vivo. Design, synthesis and biological evaluation of tanshinone Design, synthesis and biological evaluation of tanshinone IIA-based analogues:Potent inhibitors of microtubule formation and angiogenesis Eur J Med Chem the in vivo anti-angiogenic effect of 2f was confirmed via a zebrafish model test. The satisfactory physicochemical property and metabolic stability of 2f, as well as improved water
Design, synthesis, molecular modeling and anti-HIV 1 integrase activity of a series of photoactivable diketo acid-containing inhibitors as affinity probes 3 0 0 Synthesis and antidiabetic activity of novel Jul 26, 2021 · Design and synthesis of novel GCGR antagonists as biphenylsulfonamide derivatives. The compound of 7aB-3 lowering the blood glucose level in HFD-induced obese mice.
[Design, synthesis and anti-oxidative evaluation of L-amino acid prodrugs of scutellarein]. [Article in Chinese] Fu XZ(1), Zhang W, Wang YL, Lan YY, Wang AM, Zhou W, Huang Y, Li J, Xing FJ, Liu Y. Author information:(1)School of Pharmacy, Guiyang Medical College, Guiyang 550004, China.